Reset
Start Over
Help
Publication Permission Requests
Example Input Mode:
Partner Data
CBIS
Matrix
Example Data Type:
Secondary Screen (Kd)
Primary Screen(% control or competition)
If the input file contains Primary and Secondary Data, use:
Primary
Secondary
Assay Data File:
.txt or .csv format - download examples:
Bromodomain
Kd
Primary
To highlight spots, select a compound(s), click 'fill' and select entries.
Create Images for:
Vandetanib
Highlight These Spots (
fill
):
Vandetanib|ABL1-nonphosphorylated|48
Vandetanib|ABL2|69
Vandetanib|ACVR1|150
Vandetanib|ACVRL1|470
Vandetanib|ADCK3|4500
Vandetanib|ADCK4|1700
Vandetanib|ALK|2100
Vandetanib|AMPK-alpha1|3000
Vandetanib|AURKC|1500
Vandetanib|AXL|250
Vandetanib|BLK|66
Vandetanib|BMPR1B|240
Vandetanib|BRK|160
Vandetanib|BTK|1700
Vandetanib|CDK7|4100
Vandetanib|CIT|1800
Vandetanib|CSF1R|1200
Vandetanib|CSK|2500
Vandetanib|CSNK1E|3000
Vandetanib|DDR1|11
Vandetanib|DDR2|320
Vandetanib|DMPK2|2200
Vandetanib|EGFR|9.5
Vandetanib|EPHA1|230
Vandetanib|EPHA2|1100
Vandetanib|EPHA3|2000
Vandetanib|EPHA4|1600
Vandetanib|EPHA5|240
Vandetanib|EPHA6|50
Vandetanib|EPHA7|2400
Vandetanib|EPHA8|91
Vandetanib|EPHB1|290
Vandetanib|EPHB2|440
Vandetanib|EPHB4|520
Vandetanib|EPHB6|76
Vandetanib|ERBB2|2600
Vandetanib|ERBB3|160
Vandetanib|ERBB4|480
Vandetanib|ERK3|1500
Vandetanib|FGFR1|560
Vandetanib|FGFR2|1100
Vandetanib|FGFR3|1600
Vandetanib|FGFR4|2300
Vandetanib|FGR|270
Vandetanib|FLT1|260
Vandetanib|FLT3|850
Vandetanib|FLT4|1100
Vandetanib|FRK|170
Vandetanib|FYN|360
Vandetanib|GAK|86
Vandetanib|HCK|360
Vandetanib|HPK1|5500
Vandetanib|HUNK|4100
Vandetanib|IRAK1|1200
Vandetanib|IRAK4|75
Vandetanib|KIT|260
Vandetanib|LCK|17
Vandetanib|LOK|81
Vandetanib|LTK|550
Vandetanib|LYN|110
Vandetanib|MAP3K4|3000
Vandetanib|MAP4K2|1600
Vandetanib|MAP4K3|1500
Vandetanib|MAP4K4|1400
Vandetanib|MAP4K5|450
Vandetanib|MEK1|1800
Vandetanib|MEK2|1100
Vandetanib|MEK5|49
Vandetanib|MERTK|1400
Vandetanib|MET|5700
Vandetanib|MINK|3400
Vandetanib|MKNK1|360
Vandetanib|MKNK2|1700
Vandetanib|MRCKA|2600
Vandetanib|MRCKB|2500
Vandetanib|PDGFRA|230
Vandetanib|PDGFRB|88
Vandetanib|PHKG1|1100
Vandetanib|PHKG2|7900
Vandetanib|PLK4|620
Vandetanib|QSK|3900
Vandetanib|RET|34
Vandetanib|RIPK2|4.6
Vandetanib|RIPK4|620
Vandetanib|ROCK2|3600
Vandetanib|RSK1(Kin.Dom.2-C-terminal)|400
Vandetanib|RSK4(Kin.Dom.2-C-terminal)|240
Vandetanib|S6K1|1600
Vandetanib|SIK|1900
Vandetanib|SIK2|430
Vandetanib|SLK|95
Vandetanib|SRC|70
Vandetanib|SRMS|1900
Vandetanib|STK33|1400
Vandetanib|STK35|56
Vandetanib|TESK1|3700
Vandetanib|TIE1|1500
Vandetanib|TIE2|1000
Vandetanib|TNIK|2300
Vandetanib|TNNI3K|2800
Vandetanib|TXK|3700
Vandetanib|TYRO3|93
Vandetanib|ULK3|6400
Vandetanib|VEGFR2|820
Vandetanib|YANK1|5000
Vandetanib|YES|120
Vandetanib|YSK4|980
Vandetanib|ZAK|5100
Vandetanib|ABL1-nonphosphorylated
Vandetanib|ABL2
Vandetanib|ACVR1
Vandetanib|ACVRL1
Vandetanib|ADCK3
Vandetanib|ADCK4
Vandetanib|ALK
Vandetanib|AMPK-alpha1
Vandetanib|AURKC
Vandetanib|AXL
Vandetanib|BLK
Vandetanib|BMPR1B
Vandetanib|BRK
Vandetanib|BTK
Vandetanib|CDK7
Vandetanib|CIT
Vandetanib|CSF1R
Vandetanib|CSK
Vandetanib|CSNK1E
Vandetanib|DDR1
Vandetanib|DDR2
Vandetanib|DMPK2
Vandetanib|EGFR
Vandetanib|EPHA1
Vandetanib|EPHA2
Vandetanib|EPHA3
Vandetanib|EPHA4
Vandetanib|EPHA5
Vandetanib|EPHA6
Vandetanib|EPHA7
Vandetanib|EPHA8
Vandetanib|EPHB1
Vandetanib|EPHB2
Vandetanib|EPHB4
Vandetanib|EPHB6
Vandetanib|ERBB2
Vandetanib|ERBB3
Vandetanib|ERBB4
Vandetanib|ERK3
Vandetanib|FGFR1
Vandetanib|FGFR2
Vandetanib|FGFR3
Vandetanib|FGFR4
Vandetanib|FGR
Vandetanib|FLT1
Vandetanib|FLT3
Vandetanib|FLT4
Vandetanib|FRK
Vandetanib|FYN
Vandetanib|GAK
Vandetanib|HCK
Vandetanib|HPK1
Vandetanib|HUNK
Vandetanib|IRAK1
Vandetanib|IRAK4
Vandetanib|KIT
Vandetanib|LCK
Vandetanib|LOK
Vandetanib|LTK
Vandetanib|LYN
Vandetanib|MAP3K4
Vandetanib|MAP4K2
Vandetanib|MAP4K3
Vandetanib|MAP4K4
Vandetanib|MAP4K5
Vandetanib|MEK1
Vandetanib|MEK2
Vandetanib|MEK5
Vandetanib|MERTK
Vandetanib|MET
Vandetanib|MINK
Vandetanib|MKNK1
Vandetanib|MKNK2
Vandetanib|MRCKA
Vandetanib|MRCKB
Vandetanib|PDGFRA
Vandetanib|PDGFRB
Vandetanib|PHKG1
Vandetanib|PHKG2
Vandetanib|PLK4
Vandetanib|QSK
Vandetanib|RET
Vandetanib|RIPK2
Vandetanib|RIPK4
Vandetanib|ROCK2
Vandetanib|RSK1(Kin.Dom.2-C-terminal)
Vandetanib|RSK4(Kin.Dom.2-C-terminal)
Vandetanib|S6K1
Vandetanib|SIK
Vandetanib|SIK2
Vandetanib|SLK
Vandetanib|SRC
Vandetanib|SRMS
Vandetanib|STK33
Vandetanib|STK35
Vandetanib|TESK1
Vandetanib|TIE1
Vandetanib|TIE2
Vandetanib|TNIK
Vandetanib|TNNI3K
Vandetanib|TXK
Vandetanib|TYRO3
Vandetanib|ULK3
Vandetanib|VEGFR2
Vandetanib|YANK1
Vandetanib|YES
Vandetanib|YSK4
Vandetanib|ZAK
Vandetanib|ABL1-nonphosphorylated|48
Vandetanib|ABL2|69
Vandetanib|ACVR1|150
Vandetanib|ACVRL1|470
Vandetanib|ADCK3|4500
Vandetanib|ADCK4|1700
Vandetanib|ALK|2100
Vandetanib|AMPK-alpha1|3000
Vandetanib|AURKC|1500
Vandetanib|AXL|250
Vandetanib|BLK|66
Vandetanib|BMPR1B|240
Vandetanib|BRK|160
Vandetanib|BTK|1700
Vandetanib|CDK7|4100
Vandetanib|CIT|1800
Vandetanib|CSF1R|1200
Vandetanib|CSK|2500
Vandetanib|CSNK1E|3000
Vandetanib|DDR1|11
Vandetanib|DDR2|320
Vandetanib|DMPK2|2200
Vandetanib|EGFR|9.5
Vandetanib|EPHA1|230
Vandetanib|EPHA2|1100
Vandetanib|EPHA3|2000
Vandetanib|EPHA4|1600
Vandetanib|EPHA5|240
Vandetanib|EPHA6|50
Vandetanib|EPHA7|2400
Vandetanib|EPHA8|91
Vandetanib|EPHB1|290
Vandetanib|EPHB2|440
Vandetanib|EPHB4|520
Vandetanib|EPHB6|76
Vandetanib|ERBB2|2600
Vandetanib|ERBB3|160
Vandetanib|ERBB4|480
Vandetanib|ERK3|1500
Vandetanib|FGFR1|560
Vandetanib|FGFR2|1100
Vandetanib|FGFR3|1600
Vandetanib|FGFR4|2300
Vandetanib|FGR|270
Vandetanib|FLT1|260
Vandetanib|FLT3|850
Vandetanib|FLT4|1100
Vandetanib|FRK|170
Vandetanib|FYN|360
Vandetanib|GAK|86
Vandetanib|HCK|360
Vandetanib|HPK1|5500
Vandetanib|HUNK|4100
Vandetanib|IRAK1|1200
Vandetanib|IRAK4|75
Vandetanib|KIT|260
Vandetanib|LCK|17
Vandetanib|LOK|81
Vandetanib|LTK|550
Vandetanib|LYN|110
Vandetanib|MAP3K4|3000
Vandetanib|MAP4K2|1600
Vandetanib|MAP4K3|1500
Vandetanib|MAP4K4|1400
Vandetanib|MAP4K5|450
Vandetanib|MEK1|1800
Vandetanib|MEK2|1100
Vandetanib|MEK5|49
Vandetanib|MERTK|1400
Vandetanib|MET|5700
Vandetanib|MINK|3400
Vandetanib|MKNK1|360
Vandetanib|MKNK2|1700
Vandetanib|MRCKA|2600
Vandetanib|MRCKB|2500
Vandetanib|PDGFRA|230
Vandetanib|PDGFRB|88
Vandetanib|PHKG1|1100
Vandetanib|PHKG2|7900
Vandetanib|PLK4|620
Vandetanib|QSK|3900
Vandetanib|RET|34
Vandetanib|RIPK2|4.6
Vandetanib|RIPK4|620
Vandetanib|ROCK2|3600
Vandetanib|RSK1(Kin.Dom.2-C-terminal)|400
Vandetanib|RSK4(Kin.Dom.2-C-terminal)|240
Vandetanib|S6K1|1600
Vandetanib|SIK|1900
Vandetanib|SIK2|430
Vandetanib|SLK|95
Vandetanib|SRC|70
Vandetanib|SRMS|1900
Vandetanib|STK33|1400
Vandetanib|STK35|56
Vandetanib|TESK1|3700
Vandetanib|TIE1|1500
Vandetanib|TIE2|1000
Vandetanib|TNIK|2300
Vandetanib|TNNI3K|2800
Vandetanib|TXK|3700
Vandetanib|TYRO3|93
Vandetanib|ULK3|6400
Vandetanib|VEGFR2|820
Vandetanib|YANK1|5000
Vandetanib|YES|120
Vandetanib|YSK4|980
Vandetanib|ZAK|5100
clear
Select Highlight spots color from Pallette:
(also used in table view)
Tree Image Options
Restore default options
Spot options:
IndianRed
PaleGreen
Gold
PowderBlue
Fill?
Outline?
Outline thickness:
1
2
3
4
5
Select Spots Color from Pallette:
(spot highlight color below)
micro
nano
Spot Size:
Scaling Factor:
.1
.2
.3
.4
.5
.6
.7
.8
.9
1
1.1
1.2
1.3
Area increase factor:
100%
90%
80%
70%
60%
50%
(per change of 10x Kd or 10% Competition)
Legend options:
Left align Text
Right align Text
Label options:
Compound Name?
Compound Name Font:
.5
1
1.5
2
Show Assay Panel information?
Show Panel Spots?
Append Concentration? (i.e., 'AB500@1000nm'; check before loading.)
Background Image:
Target labels?
Dark Tree Branch image?
Hide Lipid, Mutant, ATypical and Pathogen?
Spot options:
Spot Color transparency level:
none
low
medium-low
medium
high
no color
Spot Cutoff Value:
Kd (nM) (Blank for no cutoff)
Spot outline only?
Format:
JPEG(200KB per image)
Publication Quality(5MB image)
Create Publication Quality (5MB bitmap) Image for:
Select Compound
Vandetanib
size/quality
100
90
80
70
60
50
40
30
% of original
White Space Border:
Yes
No
Preview and Highlighting
Highlight an assay by clicking on the spot or checking the box next to the Gene Symbol Name.
Click 'Update' to create the new images.
Compound To Highlight:
None
Vandetanib
Highlight Panel?
* WildType kinase assays appear in both the main TREEspot and Mutant kinase dendrogams.
Human Kinome image created by KINOMEscan.
2 images created. To download (copy and paste) all images to your local machine click Open/Browse Image Folder.
Images Saved To:
D:\Eurofins\PROD\Applications\FrontOffice_Discovery\StudyManagement\TreeSpot\HTSTools\TreeImages\932_3v5smmgwlxjtctitzko0iakk\
Open/Browse Image Folder
View Options:
(These options do not modify the images that have been created, only the view on this page)
Vandetanib
Legend
Show Selected
Size:
Select Size
small
medium
full size
Images per Row:
1
Legend Resize?
Hover the cursor to identify spots and click to highlighted it. To save an image click the Zoom/Download link.
Zoom/Download
Highlight
Locate an Assay
ABL1-nonphosphorylated
ABL1-nonphosphorylated
ABL2
ACVR1
ACVRL1
ADCK4
ALK
ALK
AURKC
AXL
BLK
BMPR1B
BRK
BTK
CIT
CSF1R
CSK
DDR1
DDR2
DMPK2
EGFR
EGFR
EPHA1
EPHA2
EPHA3
EPHA4
EPHA5
EPHA6
EPHA7
EPHA8
EPHB1
EPHB2
EPHB4
EPHB6
ERBB2
ERBB3
ERBB4
ERK3
FGFR1
FGFR2
FGFR3
FGFR3
FGFR4
FGR
FLT1
FLT3
FLT3
FLT4
FRK
FYN
GAK
HCK
IRAK1
IRAK4
KIT
KIT
LCK
LOK
LTK
LYN
MAP4K2
MAP4K3
MAP4K4
MAP4K5
MEK1
MEK2
MEK5
MERTK
MKNK1
MKNK2
MRCKA
MRCKB
PDGFRA
PDGFRB
PHKG1
PLK4
RET
RET
RIPK2
RIPK4
RSK1(Kin.Dom.2-C-terminal)
RSK4(Kin.Dom.2-C-terminal)
S6K1
SIK
SIK2
SLK
SRC
SRMS
STK33
STK35
TIE1
TIE2
TNIK
TNNI3K
TYRO3
VEGFR2
YES
YSK4
Legend
Data Table View:
Show All Data
Only Selected Compounds/Trees
TREE
spot
Copyright © 2005-2012 KINOMEscan, a division of DiscoveRx Corp. All Rights Reserved.